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Cat. No. Product Name Target Signaling Pathways
TQ0316 Ingenol-5,20-acetonide-3-O-angelate

Ingenol 5,20-acetonide 3-angelate,Ingenol 3-angelate 5,20-acetonide,巨大戟醇-5,20-缩丙酮-3-当归酸酯

Others Others
Ingenol-5,20-acetonide-3-O-angelate (Ingenol 5,20-acetonide 3-angelate) 是一种天然产物。
TN1047 Ingenol mebutate

Ingenol 3-Angelate,巨大戟醇甲基丁烯酸酯,PEP005

gp120/CD4; HIV Protease; PKC Chromatin/Epigenetic; Cytoskeletal Signaling; Immunology/Inflammation; Microbiology/Virology; Proteases/Proteasome
Ingenol mebutate (Ingenol 3-Angelate) 是 PKC 的有效激动剂,包括 PKC-α、PKC-β、PKC-γ、PKC-δ 和 PKC-ε,Kis 为 0.3、0.105、0.162、0.376 和 0.171 nM。 Ingenol mebutate 具有抗炎和抗肿瘤活性。
TN1049 Ingenol-5,20-acetonide

Others Others
Ingenol-5,20-acetonide 是一种天然化合物,Ingenol 3-Angelate 的类似物,当局部用于治疗光化性角化病时具有抗肿瘤活性。
TN2799 20-Deoxyingenol 3-angelate

PKC Chromatin/Epigenetic; Cytoskeletal Signaling
20-Deoxyingenol 3-angelate and ingenol 20-acetate 3-angelate are known as promoters of tumors of mouse skin. 20-Deoxyingenol 3-angelate can induce significant platelet aggregation accompanied by induction of phosphorylation of PKC substrates in platelets,

天然产物

Ingenol-5,20-acetonide-3-O-angelate
Cat.No: TQ0316
Synonym: Ingenol 5,20-acetonide 3-angelate,Ingenol 3-angelate 5,20-acetonide,巨大戟醇-5,20-缩丙酮-3-当归酸酯
Target: Others
Ingenol mebutate
Cat.No: TN1047
Synonym: Ingenol 3-Angelate,巨大戟醇甲基丁烯酸酯,PEP005
Target: gp120/CD4, HIV Protease, PKC
Ingenol-5,20-acetonide
Cat.No: TN1049
Synonym:
Target: Others
20-Deoxyingenol 3-angelate
Cat.No: TN2799
Synonym:
Target: PKC
TargetMol Loading
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